INCB018424 KINOMEscan - Dataset (ID:20173)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Ruxolitinib | DCAMKL2 | 760.0 | nM |
| Ruxolitinib | DCAMKL3 | 260.0 | nM |
| Ruxolitinib | DDR1 | nM | |
| Ruxolitinib | DDR2 | nM | |
| Ruxolitinib | M3K12 | nM | |
| Ruxolitinib | DMPK | 3500.0 | nM |
| Ruxolitinib | DMPK2 | nM | |
| Ruxolitinib | DRAK1 | 6200.0 | nM |
| Ruxolitinib | DRAK2 | 3500.0 | nM |
| Ruxolitinib | DYRK1A | 910.0 | nM |
| Ruxolitinib | DYRK1B | nM | |
| Ruxolitinib | DYRK2 | 3700.0 | nM |
| Ruxolitinib | EGFR | nM | |
| Ruxolitinib | EGFR(E746-A750del) | nM | |
| Ruxolitinib | EGFR(G719C) | nM | |
| Ruxolitinib | EGFR(G719S) | nM | |
| Ruxolitinib | EGFR(L747-E749del, A750P) | nM | |
| Ruxolitinib | EGFR(L747-S752del, P753S) | nM | |
| Ruxolitinib | EGFR(L747-T751del,Sins) | nM | |
| Ruxolitinib | EGFR(L858R) | nM | |
| Ruxolitinib | EGFR(L858R,T790M) | nM | |
| Ruxolitinib | EGFR(L861Q) | nM | |
| Ruxolitinib | EGFR(S752-I759del) | nM | |
| Ruxolitinib | EGFR(T790M) | nM | |
| Ruxolitinib | EIF2AK1 | nM |