INCB018424 KINOMEscan - Dataset (ID:20173)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | IKKB | 2300.0 | nM |
Ruxolitinib | IKKE | 1200.0 | nM |
Ruxolitinib | INSR | nM | |
Ruxolitinib | INSRR | nM | |
Ruxolitinib | IRAK1 | 290.0 | nM |
Ruxolitinib | IRAK3 | nM | |
Ruxolitinib | IRAK4 | nM | |
Ruxolitinib | ITK | nM | |
Ruxolitinib | JAK1(JH1domain-catalytic) | 3.4 | nM |
Ruxolitinib | JAK1(JH2domain-pseudokinase) | nM | |
Ruxolitinib | JAK2(JH1domain-catalytic) | 0.0 | nM |
Ruxolitinib | JAK3(JH1domain-catalytic) | 2.0 | nM |
Ruxolitinib | JNK1 | 4800.0 | nM |
Ruxolitinib | JNK3 | nM | |
Ruxolitinib | KC1G1 | nM | |
Ruxolitinib | KC1G2 | nM | |
Ruxolitinib | KCC2D | 90.0 | nM |
Ruxolitinib | KCC4 | nM | |
Ruxolitinib | KGP1 | nM | |
Ruxolitinib | KGP2 | 690.0 | nM |
Ruxolitinib | KIT | nM | |
Ruxolitinib | KIT(A829P) | 6300.0 | nM |
Ruxolitinib | KIT(D816H) | 6300.0 | nM |
Ruxolitinib | KIT(D816V) | 7100.0 | nM |
Ruxolitinib | KIT(L576P) | nM |