INCB018424 KINOMEscan - Dataset (ID:20173)

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Small Molecule Protein Kd Conc unit
Ruxolitinib AKT2
nM
Ruxolitinib AKT3
nM
Ruxolitinib ALK 1500.0
nM
Ruxolitinib AMPK-alpha1
nM
Ruxolitinib AMPK-alpha2
nM
Ruxolitinib ANKK1 390.0
nM
Ruxolitinib AURKA
nM
Ruxolitinib AURKB
nM
Ruxolitinib AURKC 8700.0
nM
Ruxolitinib AXL
nM
Ruxolitinib BIKE 210.0
nM
Ruxolitinib BLK
nM
Ruxolitinib BMPR1A
nM
Ruxolitinib BMPR1B 1800.0
nM
Ruxolitinib BMPR2 930.0
nM
Ruxolitinib BMX
nM
Ruxolitinib BRAF 2200.0
nM
Ruxolitinib BRAF(V600E) 4200.0
nM
Ruxolitinib BRSK1
nM
Ruxolitinib BRSK2
nM
Ruxolitinib BTK
nM
Ruxolitinib CAMK1 470.0
nM
Ruxolitinib CAMK1D 120.0
nM
Ruxolitinib CAMK1G 2200.0
nM
Ruxolitinib CAMK2A 46.0
nM