INCB018424 KINOMEscan - Dataset (ID:20173)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | AKT2 | nM | |
Ruxolitinib | AKT3 | nM | |
Ruxolitinib | ALK | 1500.0 | nM |
Ruxolitinib | AMPK-alpha1 | nM | |
Ruxolitinib | AMPK-alpha2 | nM | |
Ruxolitinib | ANKK1 | 390.0 | nM |
Ruxolitinib | AURKA | nM | |
Ruxolitinib | AURKB | nM | |
Ruxolitinib | AURKC | 8700.0 | nM |
Ruxolitinib | AXL | nM | |
Ruxolitinib | BIKE | 210.0 | nM |
Ruxolitinib | BLK | nM | |
Ruxolitinib | BMPR1A | nM | |
Ruxolitinib | BMPR1B | 1800.0 | nM |
Ruxolitinib | BMPR2 | 930.0 | nM |
Ruxolitinib | BMX | nM | |
Ruxolitinib | BRAF | 2200.0 | nM |
Ruxolitinib | BRAF(V600E) | 4200.0 | nM |
Ruxolitinib | BRSK1 | nM | |
Ruxolitinib | BRSK2 | nM | |
Ruxolitinib | BTK | nM | |
Ruxolitinib | CAMK1 | 470.0 | nM |
Ruxolitinib | CAMK1D | 120.0 | nM |
Ruxolitinib | CAMK1G | 2200.0 | nM |
Ruxolitinib | CAMK2A | 46.0 | nM |