INCB018424 KINOMEscan - Dataset (ID:20173)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | ULK2 | 190.0 | nM |
Ruxolitinib | PLK4 | 200.0 | nM |
Ruxolitinib | MKNK2 | 200.0 | nM |
Ruxolitinib | BIKE | 210.0 | nM |
Ruxolitinib | DCAMKL3 | 260.0 | nM |
Ruxolitinib | YSK4 | 270.0 | nM |
Ruxolitinib | RET(V804L) | 280.0 | nM |
Ruxolitinib | IRAK1 | 290.0 | nM |
Ruxolitinib | LRRK2 | 290.0 | nM |
Ruxolitinib | ULK1 | 300.0 | nM |
Ruxolitinib | TAOK2 | 310.0 | nM |
Ruxolitinib | CAMK2B | 310.0 | nM |
Ruxolitinib | SNARK | 320.0 | nM |
Ruxolitinib | TRKC | 330.0 | nM |
Ruxolitinib | RPS6KA4(Kin.Dom.2-C-terminal) | 340.0 | nM |
Ruxolitinib | TRKB | 360.0 | nM |
Ruxolitinib | MYLK | 360.0 | nM |
Ruxolitinib | ANKK1 | 390.0 | nM |
Ruxolitinib | LTK | 440.0 | nM |
Ruxolitinib | CLK2 | 460.0 | nM |
Ruxolitinib | MP2K3 | 470.0 | nM |
Ruxolitinib | CAMK1 | 470.0 | nM |
Ruxolitinib | TTK | 480.0 | nM |
Ruxolitinib | STK16 | 490.0 | nM |
Ruxolitinib | MAST1 | 520.0 | nM |