INCB018424 KINOMEscan - Dataset (ID:20173)

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Small Molecule Protein Kd Conc unit
Ruxolitinib TAK1 730.0
nM
Ruxolitinib TAOK1 1300.0
nM
Ruxolitinib TAOK2 310.0
nM
Ruxolitinib TAOK3 590.0
nM
Ruxolitinib TBK1 1700.0
nM
Ruxolitinib TEC
nM
Ruxolitinib TESK1
nM
Ruxolitinib TGFBR1
nM
Ruxolitinib TGFBR2
nM
Ruxolitinib TIE1
nM
Ruxolitinib TIE2
nM
Ruxolitinib TLK1
nM
Ruxolitinib TLK2
nM
Ruxolitinib TNIK
nM
Ruxolitinib TNK1
nM
Ruxolitinib TNK2 2600.0
nM
Ruxolitinib TNNI3K
nM
Ruxolitinib TRKA 1500.0
nM
Ruxolitinib TRKB 360.0
nM
Ruxolitinib TRKC 330.0
nM
Ruxolitinib TRPM6
nM
Ruxolitinib TSSK1
nM
Ruxolitinib TTK 480.0
nM
Ruxolitinib TXK
nM
Ruxolitinib TYK2(JH1domain-catalytic) 0.9
nM