INCB018424 KINOMEscan - Dataset (ID:20173)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Ruxolitinib | PRKX | nM | |
| Ruxolitinib | PRP4 | nM | |
| Ruxolitinib | FAK2 | nM | |
| Ruxolitinib | SIK3 | 1300.0 | nM |
| Ruxolitinib | RAF1 | nM | |
| Ruxolitinib | RET | 720.0 | nM |
| Ruxolitinib | RET(M918T) | 630.0 | nM |
| Ruxolitinib | RET(V804L) | 280.0 | nM |
| Ruxolitinib | RET(V804M) | 190.0 | nM |
| Ruxolitinib | RIOK1 | 2500.0 | nM |
| Ruxolitinib | RIOK2 | 1200.0 | nM |
| Ruxolitinib | RIOK3 | 2000.0 | nM |
| Ruxolitinib | RIPK1 | nM | |
| Ruxolitinib | RIPK2 | nM | |
| Ruxolitinib | RIPK4 | 2100.0 | nM |
| Ruxolitinib | RIPK5 | nM | |
| Ruxolitinib | ROCK1 | 60.0 | nM |
| Ruxolitinib | ROCK2 | 52.0 | nM |
| Ruxolitinib | ROS1 | nM | |
| Ruxolitinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
| Ruxolitinib | RPS6KA4(Kin.Dom.2-C-terminal) | 340.0 | nM |
| Ruxolitinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
| Ruxolitinib | RPS6KA5(Kin.Dom.2-C-terminal) | 140.0 | nM |
| Ruxolitinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
| Ruxolitinib | RSK1(Kin.Dom.2-C-terminal) | 120.0 | nM |