BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Afatinib | FES | nM | |
| Afatinib | FGFR1 | nM | |
| Afatinib | FGFR2 | nM | |
| Afatinib | FGFR3 | nM | |
| Afatinib | FGFR3(G697C) | nM | |
| Afatinib | FGFR4 | nM | |
| Afatinib | FGR | nM | |
| Afatinib | VGFR1 | nM | |
| Afatinib | FLT3 | nM | |
| Afatinib | FLT3(D835H) | 1800.0 | nM |
| Afatinib | FLT3(D835Y) | 1400.0 | nM |
| Afatinib | FLT3(ITD) | nM | |
| Afatinib | FLT3(K663Q) | nM | |
| Afatinib | FLT3(N841I) | 6200.0 | nM |
| Afatinib | FLT3(R834Q) | nM | |
| Afatinib | FLT4 | nM | |
| Afatinib | FRK | 1400.0 | nM |
| Afatinib | FYN | nM | |
| Afatinib | GAK | 79.0 | nM |
| Afatinib | GCN2(Kin.Dom.2,S808G) | nM | |
| Afatinib | GRK1 | nM | |
| Afatinib | GRK4 | nM | |
| Afatinib | GRK7 | nM | |
| Afatinib | GSK3A | nM | |
| Afatinib | GSK3B | nM |