BIBW-2992 KINOMEscan - Dataset (ID:20172)

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Small Molecule Protein Kd Conc unit
Afatinib MET(Y1235D) 2600.0
nM
Afatinib ABL1(T315I)-nonphosphorylated 2600.0
nM
Afatinib RIPK2 2700.0
nM
Afatinib SRC 2800.0
nM
Afatinib DYRK1B 2800.0
nM
Afatinib ABL1(F317I)-nonphosphorylated 2900.0
nM
Afatinib CIT 2900.0
nM
Afatinib TXK 3100.0
nM
Afatinib RSK4(Kin.Dom.2-C-terminal) 3100.0
nM
Afatinib EPHB6 3100.0
nM
Afatinib SLK 3700.0
nM
Afatinib LOK 4300.0
nM
Afatinib ERBB3 4500.0
nM
Afatinib SBK1 4800.0
nM
Afatinib AXL 5300.0
nM
Afatinib MET(M1250T) 6000.0
nM
Afatinib FLT3(N841I) 6200.0
nM
Afatinib CDC2L2
nM
Afatinib CDC2L1
nM
Afatinib ANKK1
nM
Afatinib CASK
nM
Afatinib CAMKK2
nM
Afatinib AMPK-alpha2
nM
Afatinib KKCC1
nM
Afatinib KCC4
nM