BIBW-2992 KINOMEscan - Dataset (ID:20172)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Afatinib | MKNK2 | 1600.0 | nM |
Afatinib | FRK | 1400.0 | nM |
Afatinib | FLT3(D835Y) | 1400.0 | nM |
Afatinib | ABL1-nonphosphorylated | 1300.0 | nM |
Afatinib | PHKG1 | 1300.0 | nM |
Afatinib | MP2K5 | 1300.0 | nM |
Afatinib | MK14 | 1300.0 | nM |
Afatinib | CSNK1E | 1300.0 | nM |
Afatinib | ABL1(M351T)-phosphorylated | 1200.0 | nM |
Afatinib | DYRK1A | 970.0 | nM |
Afatinib | ABL1(T315I)-phosphorylated | 870.0 | nM |
Afatinib | ABL1(Y253F)-phosphorylated | 830.0 | nM |
Afatinib | ABL1(Q252H)-nonphosphorylated | 790.0 | nM |
Afatinib | ABL1(F317I)-phosphorylated | 750.0 | nM |
Afatinib | ABL1(F317L)-nonphosphorylated | 580.0 | nM |
Afatinib | LCK | 570.0 | nM |
Afatinib | ABL1-phosphorylated | 570.0 | nM |
Afatinib | ABL1(H396P)-nonphosphorylated | 500.0 | nM |
Afatinib | ABL1(H396P)-phosphorylated | 500.0 | nM |
Afatinib | PHKG2 | 470.0 | nM |
Afatinib | ABL1(E255K)-phosphorylated | 420.0 | nM |
Afatinib | ABL1(Q252H)-phosphorylated | 380.0 | nM |
Afatinib | HIPK4 | 360.0 | nM |
Afatinib | EPHA6 | 340.0 | nM |
Afatinib | IRAK1 | 240.0 | nM |