AB-1010 KINOMEscan - Dataset (ID:20170)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Masitinib | IKKB | nM | |
Masitinib | IKKE | nM | |
Masitinib | INSR | nM | |
Masitinib | INSRR | nM | |
Masitinib | IRAK1 | nM | |
Masitinib | IRAK3 | nM | |
Masitinib | IRAK4 | nM | |
Masitinib | ITK | nM | |
Masitinib | JAK1(JH1domain-catalytic) | nM | |
Masitinib | JAK1(JH2domain-pseudokinase) | nM | |
Masitinib | JAK2(JH1domain-catalytic) | nM | |
Masitinib | JAK3(JH1domain-catalytic) | nM | |
Masitinib | JNK1 | nM | |
Masitinib | JNK3 | nM | |
Masitinib | KC1G1 | nM | |
Masitinib | KC1G2 | nM | |
Masitinib | KCC2D | nM | |
Masitinib | KCC4 | nM | |
Masitinib | KGP1 | nM | |
Masitinib | KGP2 | nM | |
Masitinib | KIT | 8.1 | nM |
Masitinib | KIT(A829P) | 12.0 | nM |
Masitinib | KIT(D816H) | 1500.0 | nM |
Masitinib | KIT(D816V) | 1300.0 | nM |
Masitinib | KIT(L576P) | 7.9 | nM |