TKI-258 KINOMEscan - Dataset (ID:20168)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Dovitinib | DCAMKL2 | nM | |
| Dovitinib | DCAMKL3 | 1300.0 | nM |
| Dovitinib | DDR1 | 2500.0 | nM |
| Dovitinib | DDR2 | 8600.0 | nM |
| Dovitinib | M3K12 | 2100.0 | nM |
| Dovitinib | DMPK | nM | |
| Dovitinib | DMPK2 | nM | |
| Dovitinib | DRAK1 | 830.0 | nM |
| Dovitinib | DRAK2 | 1800.0 | nM |
| Dovitinib | DYRK1A | nM | |
| Dovitinib | DYRK1B | nM | |
| Dovitinib | DYRK2 | 6000.0 | nM |
| Dovitinib | EGFR | nM | |
| Dovitinib | EGFR(E746-A750del) | nM | |
| Dovitinib | EGFR(G719C) | nM | |
| Dovitinib | EGFR(G719S) | nM | |
| Dovitinib | EGFR(L747-E749del, A750P) | nM | |
| Dovitinib | EGFR(L747-S752del, P753S) | nM | |
| Dovitinib | EGFR(L747-T751del,Sins) | nM | |
| Dovitinib | EGFR(L858R) | nM | |
| Dovitinib | EGFR(L858R,T790M) | 940.0 | nM |
| Dovitinib | EGFR(L861Q) | nM | |
| Dovitinib | EGFR(S752-I759del) | nM | |
| Dovitinib | EGFR(T790M) | 1400.0 | nM |
| Dovitinib | EIF2AK1 | nM |