TKI-258 KINOMEscan - Dataset (ID:20168)

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Small Molecule Protein Kd Conc unit
Dovitinib CDKL3
nM
Dovitinib CDKL5
nM
Dovitinib CHEK1 1200.0
nM
Dovitinib CHK2
nM
Dovitinib CIT 8200.0
nM
Dovitinib CLK1 6800.0
nM
Dovitinib CLK2 1700.0
nM
Dovitinib CLK3
nM
Dovitinib CLK4 6500.0
nM
Dovitinib CSF1R 60.0
nM
Dovitinib CSK
nM
Dovitinib CSNK1A1
nM
Dovitinib CSNK1A1L
nM
Dovitinib CSNK1D
nM
Dovitinib CSNK1E
nM
Dovitinib KC1G1
nM
Dovitinib KC1G2
nM
Dovitinib CSNK1G3
nM
Dovitinib CSNK2A1 2600.0
nM
Dovitinib CSNK2A2 200.0
nM
Dovitinib CTK
nM
Dovitinib DAPK1
nM
Dovitinib DAPK2
nM
Dovitinib DAPK3
nM
Dovitinib DCLK1
nM