Pazopanib KINOMEscan - Dataset (ID:20163)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pazopanib | KIT(L576P) | 1.8 | nM |
Pazopanib | PGFRB | 2.0 | nM |
Pazopanib | KIT(V559D) | 2.3 | nM |
Pazopanib | KIT | 2.8 | nM |
Pazopanib | PGFRA | 4.9 | nM |
Pazopanib | KIT(V559D,T670I) | 6.5 | nM |
Pazopanib | CSF1R | 7.9 | nM |
Pazopanib | VGFR2 | 14.0 | nM |
Pazopanib | VGFR1 | 14.0 | nM |
Pazopanib | FLT4 | 27.0 | nM |
Pazopanib | KIT(V559D,V654A) | 30.0 | nM |
Pazopanib | KIT(A829P) | 33.0 | nM |
Pazopanib | TAOK3 | 45.0 | nM |
Pazopanib | DDR1 | 57.0 | nM |
Pazopanib | EPHB6 | 81.0 | nM |
Pazopanib | LOK | 84.0 | nM |
Pazopanib | DDR2 | 98.0 | nM |
Pazopanib | TTK | 150.0 | nM |
Pazopanib | GAK | 200.0 | nM |
Pazopanib | FGFR2 | 210.0 | nM |
Pazopanib | SLK | 240.0 | nM |
Pazopanib | TAOK1 | 240.0 | nM |
Pazopanib | RIPK1 | 260.0 | nM |
Pazopanib | RET(M918T) | 270.0 | nM |
Pazopanib | PI42C | 280.0 | nM |