Pazopanib KINOMEscan - Dataset (ID:20163)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pazopanib | FLT3(R834Q) | 9600.0 | nM |
Pazopanib | BIKE | 8800.0 | nM |
Pazopanib | SIK2 | 7300.0 | nM |
Pazopanib | NEK5 | 7300.0 | nM |
Pazopanib | AURKA | 7100.0 | nM |
Pazopanib | JAK3(JH1domain-catalytic) | 6900.0 | nM |
Pazopanib | LTK | 6800.0 | nM |
Pazopanib | IRAK1 | 5900.0 | nM |
Pazopanib | RET(V804L) | 5900.0 | nM |
Pazopanib | HCK | 5700.0 | nM |
Pazopanib | YES | 5000.0 | nM |
Pazopanib | SYK | 4700.0 | nM |
Pazopanib | ABL1(F317L)-nonphosphorylated | 4400.0 | nM |
Pazopanib | NLK | 4400.0 | nM |
Pazopanib | MP2K6 | 4100.0 | nM |
Pazopanib | MARK3 | 4000.0 | nM |
Pazopanib | ABL1(T315I)-nonphosphorylated | 3800.0 | nM |
Pazopanib | CAMK1G | 3700.0 | nM |
Pazopanib | MET(M1250T) | 3400.0 | nM |
Pazopanib | TYK2(JH1domain-catalytic) | 3400.0 | nM |
Pazopanib | TIE2 | 3300.0 | nM |
Pazopanib | MERTK | 3300.0 | nM |
Pazopanib | TGFBR2 | 3000.0 | nM |
Pazopanib | MAP4K5 | 3000.0 | nM |
Pazopanib | ABL2 | 3000.0 | nM |