Erlotinib KINOMEscan - Dataset (ID:20160)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Erlotinib | DCAMKL2 | nM | |
Erlotinib | DCAMKL3 | nM | |
Erlotinib | DDR1 | 790.0 | nM |
Erlotinib | DDR2 | nM | |
Erlotinib | M3K12 | nM | |
Erlotinib | DMPK | 2900.0 | nM |
Erlotinib | DMPK2 | 3400.0 | nM |
Erlotinib | DRAK1 | 6300.0 | nM |
Erlotinib | DRAK2 | 9400.0 | nM |
Erlotinib | DYRK1A | nM | |
Erlotinib | DYRK1B | nM | |
Erlotinib | DYRK2 | 1300.0 | nM |
Erlotinib | EGFR | 0.7 | nM |
Erlotinib | EGFR(E746-A750del) | 0.5 | nM |
Erlotinib | EGFR(G719C) | 0.9 | nM |
Erlotinib | EGFR(G719S) | 0.5 | nM |
Erlotinib | EGFR(L747-E749del, A750P) | 0.5 | nM |
Erlotinib | EGFR(L747-S752del, P753S) | 0.5 | nM |
Erlotinib | EGFR(L747-T751del,Sins) | 0.4 | nM |
Erlotinib | EGFR(L858R) | 1.0 | nM |
Erlotinib | EGFR(L858R,T790M) | 190.0 | nM |
Erlotinib | EGFR(L861Q) | 1.2 | nM |
Erlotinib | EGFR(S752-I759del) | 1.6 | nM |
Erlotinib | EGFR(T790M) | 140.0 | nM |
Erlotinib | EIF2AK1 | nM |