Erlotinib KINOMEscan - Dataset (ID:20160)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Erlotinib | AAK1 | 1200.0 | nM |
| Erlotinib | ABL1(E255K)-phosphorylated | 63.0 | nM |
| Erlotinib | ABL1(F317I)-nonphosphorylated | 8200.0 | nM |
| Erlotinib | ABL1(F317I)-phosphorylated | 1100.0 | nM |
| Erlotinib | ABL1(F317L)-nonphosphorylated | 640.0 | nM |
| Erlotinib | ABL1(F317L)-phosphorylated | 150.0 | nM |
| Erlotinib | ABL1(H396P)-nonphosphorylated | 89.0 | nM |
| Erlotinib | ABL1(H396P)-phosphorylated | 58.0 | nM |
| Erlotinib | ABL1(M351T)-phosphorylated | 66.0 | nM |
| Erlotinib | ABL1(Q252H)-nonphosphorylated | 230.0 | nM |
| Erlotinib | ABL1(Q252H)-phosphorylated | 61.0 | nM |
| Erlotinib | ABL1(T315I)-nonphosphorylated | 620.0 | nM |
| Erlotinib | ABL1(T315I)-phosphorylated | 59.0 | nM |
| Erlotinib | ABL1(Y253F)-phosphorylated | 76.0 | nM |
| Erlotinib | ABL1-nonphosphorylated | 330.0 | nM |
| Erlotinib | ABL1-phosphorylated | 76.0 | nM |
| Erlotinib | ABL2 | 200.0 | nM |
| Erlotinib | ACVR1 | nM | |
| Erlotinib | ACVR1B | nM | |
| Erlotinib | ACVR2A | nM | |
| Erlotinib | ACVR2B | nM | |
| Erlotinib | ACVRL1 | nM | |
| Erlotinib | ADCK3 | 1900.0 | nM |
| Erlotinib | ADCK4 | 2500.0 | nM |
| Erlotinib | AKT1 | nM |