Erlotinib KINOMEscan - Dataset (ID:20160)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Erlotinib | ABL1(F317L)-phosphorylated | 150.0 | nM |
| Erlotinib | EGFR(L858R,T790M) | 190.0 | nM |
| Erlotinib | BLK | 190.0 | nM |
| Erlotinib | ABL2 | 200.0 | nM |
| Erlotinib | ERBB4 | 230.0 | nM |
| Erlotinib | ABL1(Q252H)-nonphosphorylated | 230.0 | nM |
| Erlotinib | LCK | 250.0 | nM |
| Erlotinib | ABL1-nonphosphorylated | 330.0 | nM |
| Erlotinib | RET(M918T) | 330.0 | nM |
| Erlotinib | FLT3(D835H) | 350.0 | nM |
| Erlotinib | EPHA6 | 440.0 | nM |
| Erlotinib | CSNK1E | 500.0 | nM |
| Erlotinib | FLT3(N841I) | 500.0 | nM |
| Erlotinib | LYN | 530.0 | nM |
| Erlotinib | TNNI3K | 570.0 | nM |
| Erlotinib | AURKC | 600.0 | nM |
| Erlotinib | ABL1(T315I)-nonphosphorylated | 620.0 | nM |
| Erlotinib | TNK1 | 630.0 | nM |
| Erlotinib | ABL1(F317L)-nonphosphorylated | 640.0 | nM |
| Erlotinib | RIPK2 | 680.0 | nM |
| Erlotinib | CIT | 680.0 | nM |
| Erlotinib | MKNK1 | 690.0 | nM |
| Erlotinib | SRC | 700.0 | nM |
| Erlotinib | JAK3(JH1domain-catalytic) | 700.0 | nM |
| Erlotinib | EPHA5 | 710.0 | nM |