Erlotinib KINOMEscan - Dataset (ID:20160)
Proteins Studied
Download: Excel (XLSX), Comma-separated (CSV)
LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200043 | M3K6 | 200043 | O95382 | Mitogen-activated protein kinase kinase kinase 6; ASK2; MAP3K6; MAPKKK6; MEKK6; MEKK6/MAP3K6; MGC125653; MGC20114 | KINOMEscan | Wild Type; Partial length | |||
200046 | AURKC | 200046 | Q9UQB9 | Aurora kinase C; AIE2; AIK3; ARK3; Aur3; AurC; AurC/Aur3; AURKC; aurora-C; STK13 | KINOMEscan | Wild Type; Full length | |||
200039 | AMPK-alpha2 | 200039 | P54646 | Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2 | KINOMEscan | Wild Type; Partial length | |||
200042 | M3K5 | 200042 | Q99683 | Mitogen-activated protein kinase kinase kinase 5; ASK; ASK/MAP3K5; ASK1; MAP3K5; MAPKKK5; MEKK5 | KINOMEscan | Wild Type; Partial length | |||
200044 | AURKA | 200044 | O14965 | Aurora kinase A; AIK; AIRK1; ARK1; Aur2; AURA; AurA/Aur2; AURKA; AURORA2; Aurora-A; Ayk1; BTAK; IAK; IAK1; MGC34538; STK15; STK6; STK7 | KINOMEscan | Wild Type; Partial length | |||
200045 | AURKB | 200045 | Q96GD4 | Aurora kinase B; AIK2; AIM1; AIM-1; ARK2; Aur1; AurB; AurB/Aur1; AURKB; aurkb-sv1; aurkb-sv2; IPL1; STK12; STK5 | KINOMEscan | Wild Type; Partial length | |||
200001 | AAK1 | 200001 | Q2M2I8 | AP2 associated kinase 1; AAK1; DKFZp686F03202; DKFZp686K16132; FLJ23712; FLJ25931; FLJ31060; FLJ42882; FLJ45252; KIAA1048; MGC138170; MGC164568; MGC164570 | KINOMEscan | Wild Type; Partial length | |||
200037 | ALK | 200037 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | Wild Type; Partial length | |||
200035 | AKT2 | 200035 | P31751 | V-akt murine thymoma viral oncogene homolog 2; AKT2; Akt2/PKBb; PKBb; PKBBETA; PRKBB; RAC-BETA | KINOMEscan | Wild Type; Partial length | |||
200041 | NUAK1 | 200041 | O60285 | NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1 | KINOMEscan | Wild Type; Partial length | |||
200036 | AKT3 | 200036 | Q9Y243 | V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2 | KINOMEscan | Wild Type; Partial length | |||
200040 | ANKK1 | 200040 | Q8NFD2 | Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288 | KINOMEscan | Wild Type; Partial length | |||
200038 | AMPK-alpha1 | 200038 | Q13131 | Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1 | KINOMEscan | Wild Type; Partial length | |||
200024 | ABL1-nonphosphorylated | 200024 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | nonphosphorylated | Wild Type; Partial length | ||
200025 | ABL1-phosphorylated | 200025 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | phosphorylated | Wild Type; Partial length | ||
200026 | ABL2 | 200026 | P42684 | V-abl Abelson murine leukemia viral oncogene homolog 2 (arg, Abelson-related gene); ABL2; ABLL; ARG; FLJ22224; FLJ31718; FLJ41441 | KINOMEscan | Wild Type; Partial length | |||
200027 | ACVR1 | 200027 | Q04771 | Activin A receptor, type I; ACTRI; ACVR1; ACVR1A; ACVRLK2; ALK2; FOP; SKR1; TSRI | KINOMEscan | Wild Type; Partial length | |||
200028 | ACVR1B | 200028 | P36896 | Activin A receptor, type IB; ACTRIB; ACVR1B; ACVRLK4; ALK4; SKR2 | KINOMEscan | Wild Type; Partial length | |||
200029 | ACVR2A | 200029 | P27037 | Activin A receptor, type IIA; ActR2; ACTRII; ACVR2; ACVR2A | KINOMEscan | Wild Type; Partial length | |||
200030 | ACVR2B | 200030 | Q13705 | Activin A receptor, type IIB; ActR2B; ACTRIIB; ActR-IIB; ACVR2B; MGC116908 | KINOMEscan | Wild Type; Partial length | |||
200031 | ACVRL1 | 200031 | P37023 | Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I | KINOMEscan | Wild Type; Partial length | |||
200032 | ADCK3 | 200032 | Q8NI60 | Chaperone, ABC1 activity of bc1 complex homolog (S. pombe); ADCK3; ARCA2; CABC1; COQ8; MGC4849; SCAR9 | KINOMEscan | Wild Type; Full length | |||
200033 | ADCK4 | 200033 | Q96D53 | AarF domain containing kinase 4; ADCK4; FLJ12229 | KINOMEscan | Wild Type; Full length | |||
200034 | AKT1 | 200034 | P31749 | V-akt murine thymoma viral oncogene homolog 1; AKT; AKT1; Akt1/PKBa; MGC99656; PKB; PKBa; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA | KINOMEscan | Wild Type; Partial length | |||
200047 | AXL | 200047 | P30530 | AXL receptor tyrosine kinase; AXL; JTK11; UFO | KINOMEscan | Wild Type; Partial length |