AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | TIE1 | 350.0 | nM |
| Barasertib | LCK | 380.0 | nM |
| Barasertib | AXL | 390.0 | nM |
| Barasertib | AURKA | 400.0 | nM |
| Barasertib | EGFR | 450.0 | nM |
| Barasertib | ERBB4 | 470.0 | nM |
| Barasertib | KIT(V559D,V654A) | 480.0 | nM |
| Barasertib | VGFR2 | 500.0 | nM |
| Barasertib | EGFR(L861Q) | 510.0 | nM |
| Barasertib | KIT(A829P) | 600.0 | nM |
| Barasertib | TAK1 | 650.0 | nM |
| Barasertib | FLT3(D835Y) | 670.0 | nM |
| Barasertib | ABL1(Q252H)-nonphosphorylated | 860.0 | nM |
| Barasertib | EGFR(L858R) | 980.0 | nM |
| Barasertib | CDC2L2 | 1000.0 | nM |
| Barasertib | ABL1(T315I)-nonphosphorylated | 1100.0 | nM |
| Barasertib | CDC2L5 | 1100.0 | nM |
| Barasertib | ABL1(H396P)-nonphosphorylated | 1200.0 | nM |
| Barasertib | MKNK2 | 1200.0 | nM |
| Barasertib | BTK | 1200.0 | nM |
| Barasertib | CDKL2 | 1200.0 | nM |
| Barasertib | CDC2L1 | 1200.0 | nM |
| Barasertib | ABL1(F317L)-nonphosphorylated | 1400.0 | nM |
| Barasertib | CSF1R | 1400.0 | nM |
| Barasertib | CHK2 | 1400.0 | nM |