AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | AAK1 | 3000.0 | nM |
| Barasertib | ABL1(E255K)-phosphorylated | 9600.0 | nM |
| Barasertib | ABL1(F317I)-nonphosphorylated | 3800.0 | nM |
| Barasertib | ABL1(F317I)-phosphorylated | 4600.0 | nM |
| Barasertib | ABL1(F317L)-nonphosphorylated | 1400.0 | nM |
| Barasertib | ABL1(F317L)-phosphorylated | 2300.0 | nM |
| Barasertib | ABL1(H396P)-nonphosphorylated | 1200.0 | nM |
| Barasertib | ABL1(H396P)-phosphorylated | nM | |
| Barasertib | ABL1(M351T)-phosphorylated | 2200.0 | nM |
| Barasertib | ABL1(Q252H)-nonphosphorylated | 860.0 | nM |
| Barasertib | ABL1(Q252H)-phosphorylated | 6800.0 | nM |
| Barasertib | ABL1(T315I)-nonphosphorylated | 1100.0 | nM |
| Barasertib | ABL1(T315I)-phosphorylated | 4800.0 | nM |
| Barasertib | ABL1(Y253F)-phosphorylated | 3800.0 | nM |
| Barasertib | ABL1-nonphosphorylated | 1500.0 | nM |
| Barasertib | ABL1-phosphorylated | 5500.0 | nM |
| Barasertib | ABL2 | nM | |
| Barasertib | ACVR1 | nM | |
| Barasertib | ACVR1B | nM | |
| Barasertib | ACVR2A | nM | |
| Barasertib | ACVR2B | nM | |
| Barasertib | ACVRL1 | nM | |
| Barasertib | ADCK3 | nM | |
| Barasertib | ADCK4 | nM | |
| Barasertib | AKT1 | nM |