AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | PRKX | nM | |
| Barasertib | PRP4 | nM | |
| Barasertib | FAK2 | nM | |
| Barasertib | SIK3 | nM | |
| Barasertib | RAF1 | nM | |
| Barasertib | RET | 80.0 | nM |
| Barasertib | RET(M918T) | 120.0 | nM |
| Barasertib | RET(V804L) | 140.0 | nM |
| Barasertib | RET(V804M) | 240.0 | nM |
| Barasertib | RIOK1 | nM | |
| Barasertib | RIOK2 | nM | |
| Barasertib | RIOK3 | nM | |
| Barasertib | RIPK1 | nM | |
| Barasertib | RIPK2 | 1800.0 | nM |
| Barasertib | RIPK4 | nM | |
| Barasertib | RIPK5 | 3000.0 | nM |
| Barasertib | ROCK1 | nM | |
| Barasertib | ROCK2 | nM | |
| Barasertib | ROS1 | nM | |
| Barasertib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
| Barasertib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
| Barasertib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
| Barasertib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
| Barasertib | RSK1(Kin.Dom.1-N-terminal) | nM | |
| Barasertib | RSK1(Kin.Dom.2-C-terminal) | nM |