AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | ANKK1 | 1500.0 | nM |
| Barasertib | ABL1-nonphosphorylated | 1500.0 | nM |
| Barasertib | EIF2AK1 | 1500.0 | nM |
| Barasertib | EGFR(T790M) | 1500.0 | nM |
| Barasertib | BLK | 1500.0 | nM |
| Barasertib | MUSK | 1500.0 | nM |
| Barasertib | LYN | 1600.0 | nM |
| Barasertib | MLTK | 1700.0 | nM |
| Barasertib | DDR1 | 1800.0 | nM |
| Barasertib | RIPK2 | 1800.0 | nM |
| Barasertib | TIE2 | 1900.0 | nM |
| Barasertib | MP2K1 | 1900.0 | nM |
| Barasertib | ABL1(M351T)-phosphorylated | 2200.0 | nM |
| Barasertib | ABL1(F317L)-phosphorylated | 2300.0 | nM |
| Barasertib | YSK4 | 2400.0 | nM |
| Barasertib | HIPK3 | 2500.0 | nM |
| Barasertib | LOK | 2800.0 | nM |
| Barasertib | S6K1 | 2800.0 | nM |
| Barasertib | KIT(D816H) | 2900.0 | nM |
| Barasertib | FLT4 | 2900.0 | nM |
| Barasertib | EGFR(L747-E749del, A750P) | 2900.0 | nM |
| Barasertib | RIPK5 | 3000.0 | nM |
| Barasertib | AAK1 | 3000.0 | nM |
| Barasertib | LTK | 3200.0 | nM |
| Barasertib | EGFR(L747-T751del,Sins) | 3500.0 | nM |