AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | ABL1(E255K)-phosphorylated | 9600.0 | nM |
| Barasertib | EGFR(L747-S752del, P753S) | 8800.0 | nM |
| Barasertib | TNIK | 8500.0 | nM |
| Barasertib | TTK | 8500.0 | nM |
| Barasertib | IRAK3 | 7900.0 | nM |
| Barasertib | SRMS | 7900.0 | nM |
| Barasertib | ABL1(Q252H)-phosphorylated | 6800.0 | nM |
| Barasertib | DDR2 | 6600.0 | nM |
| Barasertib | CDK16 | 6300.0 | nM |
| Barasertib | CDK7 | 6200.0 | nM |
| Barasertib | CIT | 5700.0 | nM |
| Barasertib | MET(Y1235D) | 5700.0 | nM |
| Barasertib | ABL1-phosphorylated | 5500.0 | nM |
| Barasertib | EGFR(S752-I759del) | 5200.0 | nM |
| Barasertib | ABL1(T315I)-phosphorylated | 4800.0 | nM |
| Barasertib | PLK4 | 4700.0 | nM |
| Barasertib | STK36 | 4600.0 | nM |
| Barasertib | ABL1(F317I)-phosphorylated | 4600.0 | nM |
| Barasertib | KIT(D816V) | 4600.0 | nM |
| Barasertib | ERBB2 | 4300.0 | nM |
| Barasertib | MP2K2 | 4200.0 | nM |
| Barasertib | HCK | 3900.0 | nM |
| Barasertib | ABL1(Y253F)-phosphorylated | 3800.0 | nM |
| Barasertib | CSK | 3800.0 | nM |
| Barasertib | ABL1(F317I)-nonphosphorylated | 3800.0 | nM |