AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | KIT | 17.0 | nM |
| Barasertib | KIT(A829P) | 600.0 | nM |
| Barasertib | KIT(D816H) | 2900.0 | nM |
| Barasertib | KIT(D816V) | 4600.0 | nM |
| Barasertib | KIT(L576P) | 34.0 | nM |
| Barasertib | KIT(V559D) | 15.0 | nM |
| Barasertib | KIT(V559D,T670I) | 7.9 | nM |
| Barasertib | KIT(V559D,V654A) | 480.0 | nM |
| Barasertib | LATS1 | nM | |
| Barasertib | LATS2 | nM | |
| Barasertib | LCK | 380.0 | nM |
| Barasertib | LIMK1 | nM | |
| Barasertib | LIMK2 | nM | |
| Barasertib | LKB1 | nM | |
| Barasertib | LOK | 2800.0 | nM |
| Barasertib | LRRK2 | nM | |
| Barasertib | LRRK2(G2019S) | nM | |
| Barasertib | LTK | 3200.0 | nM |
| Barasertib | LYN | 1600.0 | nM |
| Barasertib | M3K13 | nM | |
| Barasertib | MAK | nM | |
| Barasertib | MAP3K1 | nM | |
| Barasertib | MAP3K15 | nM | |
| Barasertib | M3K2 | nM | |
| Barasertib | MAP3K3 | nM |