AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | FES | nM | |
| Barasertib | FGFR1 | nM | |
| Barasertib | FGFR2 | nM | |
| Barasertib | FGFR3 | nM | |
| Barasertib | FGFR3(G697C) | nM | |
| Barasertib | FGFR4 | nM | |
| Barasertib | FGR | nM | |
| Barasertib | VGFR1 | 110.0 | nM |
| Barasertib | FLT3 | 8.2 | nM |
| Barasertib | FLT3(D835H) | 210.0 | nM |
| Barasertib | FLT3(D835Y) | 670.0 | nM |
| Barasertib | FLT3(ITD) | 140.0 | nM |
| Barasertib | FLT3(K663Q) | 3.9 | nM |
| Barasertib | FLT3(N841I) | 43.0 | nM |
| Barasertib | FLT3(R834Q) | 130.0 | nM |
| Barasertib | FLT4 | 2900.0 | nM |
| Barasertib | FRK | nM | |
| Barasertib | FYN | nM | |
| Barasertib | GAK | nM | |
| Barasertib | GCN2(Kin.Dom.2,S808G) | nM | |
| Barasertib | GRK1 | nM | |
| Barasertib | GRK4 | nM | |
| Barasertib | GRK7 | nM | |
| Barasertib | GSK3A | nM | |
| Barasertib | GSK3B | nM |