AZD-1152HQPA KINOMEscan-2 - Dataset (ID:20158)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Barasertib | DCAMKL2 | nM | |
| Barasertib | DCAMKL3 | nM | |
| Barasertib | DDR1 | 1800.0 | nM |
| Barasertib | DDR2 | 6600.0 | nM |
| Barasertib | M3K12 | nM | |
| Barasertib | DMPK | nM | |
| Barasertib | DMPK2 | nM | |
| Barasertib | DRAK1 | nM | |
| Barasertib | DRAK2 | nM | |
| Barasertib | DYRK1A | nM | |
| Barasertib | DYRK1B | nM | |
| Barasertib | DYRK2 | nM | |
| Barasertib | EGFR | 450.0 | nM |
| Barasertib | EGFR(E746-A750del) | nM | |
| Barasertib | EGFR(G719C) | 120.0 | nM |
| Barasertib | EGFR(G719S) | 170.0 | nM |
| Barasertib | EGFR(L747-E749del, A750P) | 2900.0 | nM |
| Barasertib | EGFR(L747-S752del, P753S) | 8800.0 | nM |
| Barasertib | EGFR(L747-T751del,Sins) | 3500.0 | nM |
| Barasertib | EGFR(L858R) | 980.0 | nM |
| Barasertib | EGFR(L858R,T790M) | nM | |
| Barasertib | EGFR(L861Q) | 510.0 | nM |
| Barasertib | EGFR(S752-I759del) | 5200.0 | nM |
| Barasertib | EGFR(T790M) | 1500.0 | nM |
| Barasertib | EIF2AK1 | 1500.0 | nM |