MLN-8054 KINOMEscan - Dataset (ID:20157)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| MLN8054 | FLT3(K663Q) | 9500.0 | nM |
| MLN8054 | DAPK2 | 9100.0 | nM |
| MLN8054 | CSK | 9000.0 | nM |
| MLN8054 | EGFR(L747-S752del, P753S) | 6400.0 | nM |
| MLN8054 | RSK1(Kin.Dom.1-N-terminal) | 4800.0 | nM |
| MLN8054 | FER | 4400.0 | nM |
| MLN8054 | DDR1 | 4200.0 | nM |
| MLN8054 | BTK | 4200.0 | nM |
| MLN8054 | LOK | 3700.0 | nM |
| MLN8054 | EPHB3 | 3500.0 | nM |
| MLN8054 | ABL2 | 3300.0 | nM |
| MLN8054 | CLK2 | 3200.0 | nM |
| MLN8054 | EGFR(L858R) | 3200.0 | nM |
| MLN8054 | FLT4 | 3100.0 | nM |
| MLN8054 | TYRO3 | 3100.0 | nM |
| MLN8054 | ROS1 | 3100.0 | nM |
| MLN8054 | BMX | 3100.0 | nM |
| MLN8054 | ABL1(T315I)-phosphorylated | 2800.0 | nM |
| MLN8054 | TNK1 | 2400.0 | nM |
| MLN8054 | FGFR1 | 2400.0 | nM |
| MLN8054 | CLK3 | 2300.0 | nM |
| MLN8054 | EPHA3 | 2100.0 | nM |
| MLN8054 | FAK2 | 2000.0 | nM |
| MLN8054 | ABL1(E255K)-phosphorylated | 1900.0 | nM |
| MLN8054 | EPHA1 | 1800.0 | nM |