MLN-8054 KINOMEscan - Dataset (ID:20157)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| MLN8054 | AURKA | 6.5 | nM |
| MLN8054 | DRAK2 | 8.1 | nM |
| MLN8054 | AURKC | 26.0 | nM |
| MLN8054 | AURKB | 43.0 | nM |
| MLN8054 | BLK | 68.0 | nM |
| MLN8054 | DRAK1 | 190.0 | nM |
| MLN8054 | FGR | 220.0 | nM |
| MLN8054 | YES | 260.0 | nM |
| MLN8054 | TIE2 | 300.0 | nM |
| MLN8054 | EPHB1 | 330.0 | nM |
| MLN8054 | EPHA2 | 370.0 | nM |
| MLN8054 | PLK4 | 410.0 | nM |
| MLN8054 | EPHA4 | 420.0 | nM |
| MLN8054 | AXL | 440.0 | nM |
| MLN8054 | ABL1(H396P)-nonphosphorylated | 510.0 | nM |
| MLN8054 | EPHB4 | 560.0 | nM |
| MLN8054 | EPHA6 | 580.0 | nM |
| MLN8054 | LCK | 590.0 | nM |
| MLN8054 | ABL1(Q252H)-nonphosphorylated | 630.0 | nM |
| MLN8054 | MERTK | 730.0 | nM |
| MLN8054 | TEC | 730.0 | nM |
| MLN8054 | ABL1(M351T)-phosphorylated | 750.0 | nM |
| MLN8054 | SRC | 800.0 | nM |
| MLN8054 | ABL1-phosphorylated | 890.0 | nM |
| MLN8054 | ABL1(H396P)-phosphorylated | 940.0 | nM |