Lapatinib KINOMEscan-2 - Dataset (ID:20155)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lapatinib | DCAMKL2 | nM | |
Lapatinib | DCAMKL3 | nM | |
Lapatinib | DDR1 | nM | |
Lapatinib | DDR2 | nM | |
Lapatinib | M3K12 | nM | |
Lapatinib | DMPK | nM | |
Lapatinib | DMPK2 | nM | |
Lapatinib | DRAK1 | nM | |
Lapatinib | DRAK2 | nM | |
Lapatinib | DYRK1A | nM | |
Lapatinib | DYRK1B | nM | |
Lapatinib | DYRK2 | nM | |
Lapatinib | EGFR | 2.4 | nM |
Lapatinib | EGFR(E746-A750del) | 8.6 | nM |
Lapatinib | EGFR(G719C) | 0.9 | nM |
Lapatinib | EGFR(G719S) | 2.1 | nM |
Lapatinib | EGFR(L747-E749del, A750P) | 2.2 | nM |
Lapatinib | EGFR(L747-S752del, P753S) | 3.9 | nM |
Lapatinib | EGFR(L747-T751del,Sins) | 3.5 | nM |
Lapatinib | EGFR(L858R) | 2.8 | nM |
Lapatinib | EGFR(L858R,T790M) | nM | |
Lapatinib | EGFR(L861Q) | 1.2 | nM |
Lapatinib | EGFR(S752-I759del) | 4.2 | nM |
Lapatinib | EGFR(T790M) | 860.0 | nM |
Lapatinib | EIF2AK1 | nM |