PLX-4720 KINOMEscan-2 - Dataset (ID:20154)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PLX-4720 | HIPK3 | 9700.0 | nM |
PLX-4720 | DCLK1 | 8100.0 | nM |
PLX-4720 | SGK3 | 7200.0 | nM |
PLX-4720 | MINK | 7100.0 | nM |
PLX-4720 | CLK1 | 6600.0 | nM |
PLX-4720 | FLT3(D835Y) | 6500.0 | nM |
PLX-4720 | FLT3(D835H) | 6100.0 | nM |
PLX-4720 | FLT3(ITD) | 6100.0 | nM |
PLX-4720 | KIT(A829P) | 5800.0 | nM |
PLX-4720 | ABL1(F317L)-phosphorylated | 5700.0 | nM |
PLX-4720 | HIPK1 | 5500.0 | nM |
PLX-4720 | HIPK4 | 5400.0 | nM |
PLX-4720 | FGFR1 | 5300.0 | nM |
PLX-4720 | RIPK1 | 5100.0 | nM |
PLX-4720 | SLK | 5100.0 | nM |
PLX-4720 | NEK2 | 5000.0 | nM |
PLX-4720 | ABL1(F317I)-phosphorylated | 5000.0 | nM |
PLX-4720 | ABL1(H396P)-phosphorylated | 5000.0 | nM |
PLX-4720 | HIPK2 | 5000.0 | nM |
PLX-4720 | KIT(V559D,V654A) | 4800.0 | nM |
PLX-4720 | SRC | 4700.0 | nM |
PLX-4720 | ABL1(E255K)-phosphorylated | 4500.0 | nM |
PLX-4720 | DDR2 | 4100.0 | nM |
PLX-4720 | KC1G2 | 4100.0 | nM |
PLX-4720 | ABL1(Q252H)-phosphorylated | 4000.0 | nM |