PLX-4720 KINOMEscan-2 - Dataset (ID:20154)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PLX-4720 | MP2K5 | 0.2 | nM |
PLX-4720 | PFCDPK1(P.falciparum) | 1.7 | nM |
PLX-4720 | SRMS | 21.0 | nM |
PLX-4720 | KIT(V559D) | 38.0 | nM |
PLX-4720 | MLTK | 41.0 | nM |
PLX-4720 | PTK6 | 48.0 | nM |
PLX-4720 | FGR | 62.0 | nM |
PLX-4720 | BRAF(V600E) | 100.0 | nM |
PLX-4720 | RAF1 | 170.0 | nM |
PLX-4720 | KIT | 180.0 | nM |
PLX-4720 | MP2K4 | 190.0 | nM |
PLX-4720 | PGFRA | 190.0 | nM |
PLX-4720 | NEK11 | 190.0 | nM |
PLX-4720 | ABL1(Q252H)-nonphosphorylated | 200.0 | nM |
PLX-4720 | PGFRB | 200.0 | nM |
PLX-4720 | BRAF | 330.0 | nM |
PLX-4720 | KIT(L576P) | 400.0 | nM |
PLX-4720 | RIPK2 | 430.0 | nM |
PLX-4720 | ABL1-nonphosphorylated | 460.0 | nM |
PLX-4720 | ABL1(H396P)-nonphosphorylated | 510.0 | nM |
PLX-4720 | SIK1 | 520.0 | nM |
PLX-4720 | MP2K1 | 550.0 | nM |
PLX-4720 | LIMK2 | 620.0 | nM |
PLX-4720 | CDK11 | 700.0 | nM |
PLX-4720 | RIOK2 | 770.0 | nM |