GDC-0941 KINOMEscan-2 - Dataset (ID:20152)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pictilisib | ICK | 9300.0 | nM |
Pictilisib | AAK1 | 9100.0 | nM |
Pictilisib | DYRK2 | 7600.0 | nM |
Pictilisib | CAMK1G | 6800.0 | nM |
Pictilisib | MELK | 5700.0 | nM |
Pictilisib | RSK4(Kin.Dom.1-N-terminal) | 5400.0 | nM |
Pictilisib | HIPK4 | 5000.0 | nM |
Pictilisib | CAMK1 | 4700.0 | nM |
Pictilisib | PCTK3 | 4600.0 | nM |
Pictilisib | TTK | 4300.0 | nM |
Pictilisib | YSK4 | 4000.0 | nM |
Pictilisib | DAPK1 | 4000.0 | nM |
Pictilisib | FLT3(N841I) | 3900.0 | nM |
Pictilisib | DYRK1B | 3800.0 | nM |
Pictilisib | RSK2(Kin.Dom.1-N-terminal) | 3000.0 | nM |
Pictilisib | GAK | 2700.0 | nM |
Pictilisib | PLK4 | 2600.0 | nM |
Pictilisib | FLT3 | 2600.0 | nM |
Pictilisib | FLT3(K663Q) | 2600.0 | nM |
Pictilisib | CSNK2A2 | 2400.0 | nM |
Pictilisib | FLT3(ITD) | 2200.0 | nM |
Pictilisib | TYK2(JH2domain-pseudokinase) | 1800.0 | nM |
Pictilisib | MK09 | 1800.0 | nM |
Pictilisib | DAPK3 | 1800.0 | nM |
Pictilisib | FLT3(D835H) | 1700.0 | nM |