GDC-0941 KINOMEscan-2 - Dataset (ID:20152)

Filter results: >>>>
  • Page 1 of 18
  • 1 to 25 of 442 records
Small Molecule Protein Kd Conc unit
Pictilisib ICK 9300.0
nM
Pictilisib AAK1 9100.0
nM
Pictilisib DYRK2 7600.0
nM
Pictilisib CAMK1G 6800.0
nM
Pictilisib MELK 5700.0
nM
Pictilisib RSK4(Kin.Dom.1-N-terminal) 5400.0
nM
Pictilisib HIPK4 5000.0
nM
Pictilisib CAMK1 4700.0
nM
Pictilisib PCTK3 4600.0
nM
Pictilisib TTK 4300.0
nM
Pictilisib YSK4 4000.0
nM
Pictilisib DAPK1 4000.0
nM
Pictilisib FLT3(N841I) 3900.0
nM
Pictilisib DYRK1B 3800.0
nM
Pictilisib RSK2(Kin.Dom.1-N-terminal) 3000.0
nM
Pictilisib GAK 2700.0
nM
Pictilisib PLK4 2600.0
nM
Pictilisib FLT3 2600.0
nM
Pictilisib FLT3(K663Q) 2600.0
nM
Pictilisib CSNK2A2 2400.0
nM
Pictilisib FLT3(ITD) 2200.0
nM
Pictilisib TYK2(JH2domain-pseudokinase) 1800.0
nM
Pictilisib MK09 1800.0
nM
Pictilisib DAPK3 1800.0
nM
Pictilisib FLT3(D835H) 1700.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records