GDC-0941 KINOMEscan-2 - Dataset (ID:20152)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Pictilisib | PIK3CA(E545A) | 0.9 | nM |
| Pictilisib | PIK3CA | 1.1 | nM |
| Pictilisib | PIK3CA(E545K) | 1.2 | nM |
| Pictilisib | PIK3CA(E542K) | 1.5 | nM |
| Pictilisib | PIK3CA(C420R) | 1.5 | nM |
| Pictilisib | PIK3CA(Q546K) | 1.7 | nM |
| Pictilisib | PIK3CA(H1047L) | 3.7 | nM |
| Pictilisib | PIK3CA(H1047Y) | 4.1 | nM |
| Pictilisib | PIK3CA(M1043I) | 4.5 | nM |
| Pictilisib | PIK3CD | 5.0 | nM |
| Pictilisib | PIK3CA(I800L) | 7.1 | nM |
| Pictilisib | PIK3CB | 16.0 | nM |
| Pictilisib | PIK3CG | 48.0 | nM |
| Pictilisib | PIK3C2B | 130.0 | nM |
| Pictilisib | MTOR | 200.0 | nM |
| Pictilisib | PIK3C2G | 300.0 | nM |
| Pictilisib | JAK1(JH2domain-pseudokinase) | 430.0 | nM |
| Pictilisib | HIPK2 | 520.0 | nM |
| Pictilisib | JNK3 | 560.0 | nM |
| Pictilisib | HIPK3 | 600.0 | nM |
| Pictilisib | CLK2 | 600.0 | nM |
| Pictilisib | RIOK2 | 670.0 | nM |
| Pictilisib | FLT3(D835Y) | 710.0 | nM |
| Pictilisib | MYLK4 | 780.0 | nM |
| Pictilisib | HIPK1 | 1100.0 | nM |