BIRB-796 KINOMEscan - Dataset (ID:20151)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Doramapimod | EPHA1 | 9800.0 | nM |
| Doramapimod | MRCKA | 9400.0 | nM |
| Doramapimod | JNK1 | 9100.0 | nM |
| Doramapimod | EGFR(G719S) | 9100.0 | nM |
| Doramapimod | ABL1(Y253F)-phosphorylated | 8500.0 | nM |
| Doramapimod | CSF1R | 8100.0 | nM |
| Doramapimod | EGFR(S752-I759del) | 7600.0 | nM |
| Doramapimod | FLT4 | 7100.0 | nM |
| Doramapimod | FAK1 | 7100.0 | nM |
| Doramapimod | EGFR | 7000.0 | nM |
| Doramapimod | EGFR(L747-T751del,Sins) | 6800.0 | nM |
| Doramapimod | MKNK1 | 6300.0 | nM |
| Doramapimod | EPHA2 | 6200.0 | nM |
| Doramapimod | EGFR(G719C) | 6000.0 | nM |
| Doramapimod | RIPK2 | 5800.0 | nM |
| Doramapimod | EGFR(L747-E749del, A750P) | 5300.0 | nM |
| Doramapimod | FLT3(N841I) | 5000.0 | nM |
| Doramapimod | ABL1(F317I)-nonphosphorylated | 4900.0 | nM |
| Doramapimod | YES | 4900.0 | nM |
| Doramapimod | EPHB1 | 4900.0 | nM |
| Doramapimod | FGFR1 | 4300.0 | nM |
| Doramapimod | VGFR2 | 3900.0 | nM |
| Doramapimod | MERTK | 3700.0 | nM |
| Doramapimod | TTK | 3300.0 | nM |
| Doramapimod | ABL1(H396P)-nonphosphorylated | 3300.0 | nM |