BIRB-796 KINOMEscan - Dataset (ID:20151)

The small molecule associated with this KINOMEscan dataset was erroneously assigned as HMS LINCS ID 10044-101 at the time of data release. The assignment was corrected to HMS LINCS 10169-999 on 2016-06-03.

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Small Molecule Protein Kd Conc unit
Doramapimod MK14 0.5
nM
Doramapimod DDR1 1.9
nM
Doramapimod MK12 2.9
nM
Doramapimod MK11 7.2
nM
Doramapimod MK09 7.3
nM
Doramapimod TIE1 8.3
nM
Doramapimod LOK 12.0
nM
Doramapimod TIE2 20.0
nM
Doramapimod DDR2 33.0
nM
Doramapimod ABL1(T315I)-nonphosphorylated 59.0
nM
Doramapimod MK13 78.0
nM
Doramapimod MAP4K4 90.0
nM
Doramapimod JNK3 110.0
nM
Doramapimod TNIK 140.0
nM
Doramapimod SLK 150.0
nM
Doramapimod TAK1 150.0
nM
Doramapimod KIT 170.0
nM
Doramapimod TRKC 190.0
nM
Doramapimod CDK11 200.0
nM
Doramapimod CDK8 220.0
nM
Doramapimod KIT(V559D) 230.0
nM
Doramapimod RET(M918T) 240.0
nM
Doramapimod KIT(L576P) 260.0
nM
Doramapimod KIT(V559D,T670I) 260.0
nM
Doramapimod EPHA8 270.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records