BIRB-796 KINOMEscan - Dataset (ID:20151)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Doramapimod | MK14 | 0.5 | nM |
Doramapimod | DDR1 | 1.9 | nM |
Doramapimod | MK12 | 2.9 | nM |
Doramapimod | MK11 | 7.2 | nM |
Doramapimod | MK09 | 7.3 | nM |
Doramapimod | TIE1 | 8.3 | nM |
Doramapimod | LOK | 12.0 | nM |
Doramapimod | TIE2 | 20.0 | nM |
Doramapimod | DDR2 | 33.0 | nM |
Doramapimod | ABL1(T315I)-nonphosphorylated | 59.0 | nM |
Doramapimod | MK13 | 78.0 | nM |
Doramapimod | MAP4K4 | 90.0 | nM |
Doramapimod | JNK3 | 110.0 | nM |
Doramapimod | TNIK | 140.0 | nM |
Doramapimod | SLK | 150.0 | nM |
Doramapimod | TAK1 | 150.0 | nM |
Doramapimod | KIT | 170.0 | nM |
Doramapimod | TRKC | 190.0 | nM |
Doramapimod | CDK11 | 200.0 | nM |
Doramapimod | CDK8 | 220.0 | nM |
Doramapimod | KIT(V559D) | 230.0 | nM |
Doramapimod | RET(M918T) | 240.0 | nM |
Doramapimod | KIT(L576P) | 260.0 | nM |
Doramapimod | KIT(V559D,T670I) | 260.0 | nM |
Doramapimod | EPHA8 | 270.0 | nM |