Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)

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Small Molecule Cell Line Drug Concentration Conc Units Timepoint Timepoint Units Measured pERK (Alexa 488) Measured p-Rb (Alexa 568) Alexa Fluor 647 Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) Image
Gefitinib AU565
0 (control)
6
hr
286.03 62.73
p-Akt
29.07 image if available
Gefitinib AU565
0 (control)
24
hr
659.08 130.41
p-Akt
134.35 image if available
Torkinib AU565
0 (control)
6
hr
228.66 55.93
p-Akt
26.38 image if available
Torkinib AU565
0 (control)
24
hr
522.19 120.45
p-Akt
94.97 image if available
GSK1059615 AU565
0 (control)
6
hr
264.31 61.82
p-Akt
28.75 image if available
GSK1059615 AU565
0 (control)
24
hr
452.11 110.23
p-Akt
88.09 image if available
MK2206 AU565
0 (control)
6
hr
215.16 63.34
p-Akt
22.81 image if available
MK2206 AU565
0 (control)
24
hr
427.04 124.23
p-Akt
78.88 image if available
Triciribine AU565
0 (control)
6
hr
231.71 61.01
p-Akt
21.54 image if available
Triciribine AU565
0 (control)
24
hr
511.74 118.54
p-Akt
102.35 image if available
Dactolisib AU565
0 (control)
6
hr
235.49 54.01
p-Akt
23.90 image if available
Dactolisib AU565
0 (control)
24
hr
496.14 121.03
p-Akt
137.91 image if available
Gefitinib HCC1954
0 (control)
6
hr
411.80 93.54
p-Akt
46.61 image if available
Gefitinib HCC1954
0 (control)
24
hr
342.49 120.54
p-Akt
84.26 image if available
Torkinib HCC1954
0 (control)
6
hr
182.67 40.88
p-Akt
23.74 image if available
Torkinib HCC1954
0 (control)
24
hr
309.60 109.35
p-Akt
76.75 image if available
GSK1059615 HCC1954
0 (control)
6
hr
241.24 67.17
p-Akt
30.76 image if available
GSK1059615 HCC1954
0 (control)
24
hr
302.50 106.62
p-Akt
73.55 image if available
MK2206 HCC1954
0 (control)
6
hr
271.78 84.99
p-Akt
42.06 image if available
MK2206 HCC1954
0 (control)
24
hr
288.09 111.00
p-Akt
78.02 image if available
Triciribine HCC1954
0 (control)
6
hr
225.27 70.45
p-Akt
36.85 image if available
Triciribine HCC1954
0 (control)
24
hr
282.25 98.69
p-Akt
60.55 image if available
Dactolisib HCC1954
0 (control)
6
hr
262.96 93.99
p-Akt
56.53 image if available
Dactolisib HCC1954
0 (control)
24
hr
357.28 117.27
p-Akt
79.92 image if available
Gefitinib MCF 10A
0 (control)
6
hr
488.10 165.19
p-Akt
54.11 image if available
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