NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | -4.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | -24.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | 28.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | MASTL | LYAVkVVK | Lys1 | -52.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 4.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | -27.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -11.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -68.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | MK14 | QELNkTIWEVPER | Other | -19.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MK14 | QELNkTIWEVPER | Other | -24.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | PAN3 | VMDPTkILITGK | -19.2 | 10 | uM | |
| NPK76-II-72-1 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | 47.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 52.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | PIK3CG | KkPLWLEFK | ATP | -2.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | -31.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | ROCK1 | kLQLELNQER | Other | 4.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | RON | IQCAIkSLSR | Lys1 | -1.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 14.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | -26.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -31.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -35.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 65.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | 11.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CK2a2 | DVkPHNVMIDHQQK | Lys2 | 18.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -79.9 | 10 | uM |