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CH5424802 KiNativ -- single dose experiment
- Dataset (ID:20105)
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Small Molecules Studied
Cell Lines Studied
Proteins Studied
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Small molecules
Cells
Proteins
10201:CH5424802
50061:HeLa
200633:ABL,ARG
200634:ABL,ARG
200635:ACK
200636:AGK
200638:AKT2,AKT3
200639:AMPKa1,AMPKa2
200640:AMPKa1,AMPKa2
200641:ARAF
200643:ATR
200644:AurA
200645:AurA,AurB,AurC
200647:BRAF
200649:KCC2D
200650:CaMK2g
200651:CaMK2g
200652:CaMKK2
200653:CASK
200654:CDC2
200655:CDK10
200656:CDK11,CDK8
200657:CDK2
200658:CDK2
200660:CDK5
200661:CDK5
200663:CDK7
200664:CDK9
200666:CHK2
200667:KC1A
200668:CK1d,CK1e
200669:CSK
200670:CSK
200672:DNAPK
200673:DNAPK
200674:DNAPK
200677:eEF2K
200678:EGFR
200679:EPHA2
200681:MK03
200682:Erk5
200683:FAK
200684:FER
200685:FER
200686:FER
200687:FYN,SRC,YES
200688:GCK
200689:GCK
200691:GCN2_domain2
200693:GSK3A
200694:GSK3B
200695:IKKA
200696:IKKB
200697:IKKE,TBK1
200698:ILK
200699:ILK
200700:IRAK1
200701:IRAK4
200702:IRE1
200703:ITPK1
200704:JAK1
200705:JAK1_domain2
200706:JAK1_domain2
200707:JNK1,JNK2,JNK3
200708:KHS1
200709:KHS1
200710:KHS1
200711:LATS1
200714:LOK
200716:LOK
200718:MAP2K1
200719:MAP2K1,MAP2K2
200720:MAP2K1,MAP2K2
200724:MAP2K4
200726:MAP2K6
200727:MAP2K6
200728:MAP2K6
200729:MP2K7
200731:M3K2
200732:M3K2,MAP3K3
200734:MAP3K4
200735:MAP3K5,MAP3K6,MAP3K7
200736:MAP3K7,TAK1
200738:MARK2
200739:MARK2,MARK3
200740:MARK3
200741:MAST1,MAST2
200743:MAST3
200744:MASTL
200745:MASTL
200746:MLK3
200747:MLKL
200748:MPSK1
200749:MSK1,MSK2_domain1
200750:MSK1_domain1
200751:MST1
200752:MST1
200753:MST1,MST2
200754:MST1,MST2
200755:MST2
200756:MST3
200757:MST3
200758:MST3,MST4,YSK1
200759:MST4,YSK1
200760:NDR1
200761:NDR1
200762:NDR1
200763:NDR1,NDR2
200764:NDR2
200767:NEK1
200768:NEK6,NEK7
200770:NEK7
200772:NEK9
200773:NEK9
200774:NEK9
200776:OSR1
200777:p38d,p38g
200778:KS6B1
200779:KS6B1
200780:p70S6K,p70S6Kb
200782:KS6B2
200784:PCTAIRE2
200785:PCTAIRE2,PCTAIRE3
200788:PHKg2
200789:PI4KA,PI4KAP2
200791:PI4KB
200793:PIK3C3
200794:PIK3CA
200795:PIK3CB
200797:PIP4K2A
200798:PI42C
200799:PI42C
200800:FYV1
200801:PITSLRE
200802:PKCa,PKCb
200805:PKD1,PKD2
200806:PKD2
200807:PKD3
200808:PKN2
200809:PKR
200810:PLK1
200812:PRPK
200814:ROCK1,ROCK2
200815:RSK1,RSK2,RSK3_domain1
200816:RSK1,RSK2_domain1
200817:RSK1_domain1
200819:RSK1_domain2
200820:RSK2_domain1
200821:RSK2_domain2
200822:RSK2_domain2
200825:RSKL1_domain1
200826:SGK3
200827:SLK
200828:SLK
200829:SLK
200830:SMG1
200834:TAO1,TAOK3
200835:TAOK2
200836:TBK1
200837:TLK1
200838:TLK2
200839:ULK3
200840:VRK2
200841:WEE1
200842:Wnk1,Wnk2,Wnk3
200843:Wnk1,Wnk2,Wnk4
200845:MLTK
200847:ZC1/HGK,ZC2/TNIK,ZC3/MINK
200872:AMPKa1
200875:ATR
200879:BRAF
200882:CAMK1D
200885:KKCC1
200888:CDC2
200890:CDK5
200894:CHK1
200896:CHK2
200904:CRK7
200907:DGKA
200908:DNAPK
200911:EPHB4
200913:Erk4
200920:FGR
200921:FRAP1
200923:GCK
200925:HGK (ZC1)
200931:IKKB
200932:IKKB
200934:ILK
200938:LATS2
200939:LOK
200940:LYN
200942:MAP2K4
200943:M3K2
200944:MAP3K5
200950:MASTL
200951:MET
200954:MST1,MST2
200958:MST4
200959:MST4,YSK1
200961:NEK4
200963:NEK6,NEK7
200964:OSR1
200965:p38a
200967:MK14
200969:PAN3
200973:PEK
200975:PIK3C2B
200979:PIK4CB
200982:PIP4K2B
200989:PKN1
200990:PKR
200992:PLK1
200996:PRP4
201002:ROCK1
201013:SRPK1
201016:STLK6
201026:ULK3
201027:YANK3
201029:ATR
201030:AurA
201033:CDK2
201034:CLK3
201035:EGFR
201036:JAK1 domain2
201037:LATS2
201038:MAP2K3
201039:MARK1
201040:NUAK1
201041:KPCI
201042:PLK1
201043:PRP4
201045:RSK1 domain1
201100:EGFR
201101:EGFR
201102:PLK1
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226 to 235 of 235 records
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Small Molecule
Cell Line
Protein
Sequence
Labeling Site
% Inhibition
Assay compound conc
Conc unit
CH5424802
HeLa
MAP2K3
MCDFGISGYLVDSVAkTMDAGCKPYMAPER
Activation Loop
5.2
10
uM
CH5424802
HeLa
MARK1
EVAVkIIDKTQLNPTSLQK
Lys1
4.7
10
uM
CH5424802
HeLa
NUAK1
VVAIkSIR
Lys1
5.2
10
uM
CH5424802
HeLa
KPCI
IYAMkVVK
Lys1
13.4
10
uM
CH5424802
HeLa
PLK1
EVFAGkIVPK
Lys1
0.5
10
uM
CH5424802
HeLa
PRP4
CNILHADIkPDNILVNESK
Lys2
20.9
10
uM
CH5424802
HeLa
RSK1 domain1
DLKPENILLDEEGHIkLTDFGLSKEAIDHEK
Lys2
76.9
10
uM
CH5424802
HeLa
EGFR
LLGAEEKEYHAEGGkVPIKWMALESILHR
Activation Loop
3.4
10
uM
CH5424802
HeLa
EGFR
GLWIPEGEKVKIPVAIkELR
Lys1
-1.4
10
uM
CH5424802
HeLa
PLK1
VIHRDLkLGNLFLNEDLEVK
Lys2
-8.9
10
uM
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