NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 CDK9
DMkAANVLITR
Lys2
28.3
 0.50
uM
NVP-BHG712 PC-3 CHK1
LSkGDGLEFK
Other
21.9
 0.50
uM
NVP-BHG712 PC-3 CHK2
VAIkIISK
Lys1
4.3
 0.50
uM
NVP-BHG712 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
9.0
 0.50
uM
NVP-BHG712 PC-3 KC1A
DIkPDNFLMGIGR
Lys2
15.1
 0.50
uM
NVP-BHG712 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
1.4
 0.50
uM
NVP-BHG712 PC-3 CSK
VSDFGLTkEASSTQDTGK
Activation Loop
2.4
 0.50
uM
NVP-BHG712 PC-3 DGKH
ATFSFCVSPLLVFVNSkSGDNQGVK
ATP
-67.0
 0.50
uM
NVP-BHG712 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
32.7
 0.50
uM
NVP-BHG712 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
-7.6
 0.50
uM
NVP-BHG712 PC-3 eEF2K
YIkYNSNSGFVR
ATP
8.1
 0.50
uM
NVP-BHG712 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
12.0
 0.50
uM
NVP-BHG712 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-17.6
 0.50
uM
NVP-BHG712 PC-3 EGFR
IPVAIkELR
Lys1
7.8
 0.50
uM
NVP-BHG712 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
70.3
 0.50
uM
NVP-BHG712 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
97.0
 0.50
uM
NVP-BHG712 PC-3 EPHA2
EVPVAIkTLK
Lys1
85.2
 0.50
uM
NVP-BHG712 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-6.7
 0.50
uM
NVP-BHG712 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
92.0
 0.50
uM
NVP-BHG712 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
94.1
 0.50
uM
NVP-BHG712 PC-3 MK03
YIHSANVLHRDLkPSNLLINTTCDLK
Lys2
-32.3
 0.50
uM
NVP-BHG712 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
11.4
 0.50
uM
NVP-BHG712 PC-3 MK01
YIHSANVLHRDLkPSNLLLNTTCDLK
Lys2
-30.5
 0.50
uM
NVP-BHG712 PC-3 Erk5
DLkPSNLLVNENCELK
Lys2
-14.3
 0.50
uM
NVP-BHG712 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
-6.8
 0.50
uM