NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | CDK14 | LVALkVIR | Lys1 | -9.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | CDK14 | DLkPQNLLISDTGELK | Lys2 | 11.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PHKg1 | DLkPENILLDDNMNIK | Lys2 | 16.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -5.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 36.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PI4KB | VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPAR | ATP | 39.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PIK3C3 | TEDGGKYPVIFkHGDDLRQDQLILQIISLMDK | ATP | 36.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 30.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | 37.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PIP4K2A | AKELPTLkDNDFINEGQK | ATP | 12.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PIP4K2B | DLPTFkDNDFLNEGQK | ATP | 21.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PI42C | VKELPTLkDMDFLNK | ATP | 20.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 8.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 12.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | FYV1 | GGkSGAAFYATEDDRFILK | ATP | 91.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | -0.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PRKACB | DLkPENLLIDHQGYIQ | Lys2 | -10.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PKD3 | NIVHCDLkPENVLLASAEPFPQVK | Lys2 | -33.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PKN1 | VLLSEFRPSGELFAIkALK | Lys1 | -11.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PKN2 | DLkLDNLLLDTEGFVK | Lys2 | -5.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PKR | DLkPSNIFLVDTK | Lys2 | 12.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PLK1 | CFEISDADTKEVFAGkIVPK | Lys1 | 3.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 10.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -1.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | 24.0 | 5.00 | uM |