NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 6.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | 7.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAP3K5,MAP3K6 | IAIkEIPER | Lys1 | -6.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 13.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | -18.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | -21.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MARK3 | EVAIkIIDKTQLNPTSLQK | Lys1 | -19.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | -27.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAST1,MAST2 | DLkPDNLLITSMGHIK | Lys2 | -10.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | 5.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | -20.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MASTL | GAFGkVYLGQK | ATP Loop | 7.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 54.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MLK1,MLKL | DLkSSNILILQK | Lys2 | -8.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 17.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MLK4 | DLkSSNILLLEK | Lys2 | 9.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MLKL | APVAIkVFK | Lys1 | 3.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 17.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | -3.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MSK1 domain1 | LGIIYRDIkLENILLDSNGHVVLTDFGLSK | Lys2 | 10.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -18.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 7.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MSK2 domain1 | DLkLENVLLDSEGHIVLTDFGLSK | Lys2 | -13.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | -8.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | 3.9 | 5.00 | uM |