NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 FER
QEDGGVYSSSGLkQIPIK
Activation Loop
11.4
 0.50
uM
NVP-BHG712 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
-26.8
 0.50
uM
NVP-BHG712 PC-3 FRAP1
IQSIAPSLQVITSkQRPR
ATP
-17.5
 0.50
uM
NVP-BHG712 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
30.9
 0.50
uM
NVP-BHG712 PC-3 GCK
DTVTSELAAVkIVK
Lys1
5.5
 0.50
uM
NVP-BHG712 PC-3 GCK
DIkGANLLLTLQGDVK
Lys2
5.1
 0.50
uM
NVP-BHG712 PC-3 GCN2_domain2
VQNKLDGCCYAVkR
Lys1
16.7
 0.50
uM
NVP-BHG712 PC-3 GCN2
LDGCCYAVkR
Lys1
13.9
 0.50
uM
NVP-BHG712 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
3.1
 0.50
uM
NVP-BHG712 PC-3 GSK3A
DIkPQNLLVDPDTAVLK
Lys2
9.7
 0.50
uM
NVP-BHG712 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
8.7
 0.50
uM
NVP-BHG712 PC-3 ERBB2
GIWIPDGENVKIPVAIkVLR
Lys1
-10.5
 0.50
uM
NVP-BHG712 PC-3 IKKA
DLkPENIVLQDVGGK
Lys2
19.4
 0.50
uM
NVP-BHG712 PC-3 IKKB
DLkPENIVLQQGEQR
Lys2
8.8
 0.50
uM
NVP-BHG712 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
-6.5
 0.50
uM
NVP-BHG712 PC-3 ILK
WQGNDIVVkVLK
Lys1
-4.2
 0.50
uM
NVP-BHG712 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
7.7
 0.50
uM
NVP-BHG712 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
-14.9
 0.50
uM
NVP-BHG712 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
10.3
 0.50
uM
NVP-BHG712 PC-3 IRE1
DLkPHNILISMPNAHGK
Lys2
-3.4
 0.50
uM
NVP-BHG712 PC-3 ITPK1
ESIFFNSHNVSkPESSSVLTELDKIEGVFERPSDEVIR
ATP
-5.2
 0.50
uM
NVP-BHG712 PC-3 JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-24.7
 0.50
uM
NVP-BHG712 PC-3 JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
10.4
 0.50
uM
NVP-BHG712 PC-3 JAK1 domain2
IGDFGLTkAIETDKEYYTVKDDR
Activation Loop
14.8
 0.50
uM
NVP-BHG712 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
4.8
 0.50
uM