XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | PC-3 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | 0.5 | 10 | uM |
| XMD-12 | HeLa | LATS1 | ALYATkTLR | Lys1 | -36.0 | 10 | uM |
| XMD-12 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 1.9 | 10 | uM |
| XMD-12 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -6.7 | 10 | uM |
| XMD-12 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 85.4 | 10 | uM |
| XMD-12 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -13.9 | 10 | uM |
| XMD-12 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 15.0 | 10 | uM |
| XMD-12 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 28.6 | 10 | uM |
| XMD-12 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | 39.1 | 10 | uM |
| XMD-12 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 28.9 | 10 | uM |
| XMD-12 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 52.3 | 10 | uM |
| XMD-12 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -23.3 | 10 | uM |
| XMD-12 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -0.6 | 10 | uM |
| XMD-12 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | 39.6 | 10 | uM |
| XMD-12 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 18.0 | 10 | uM |
| XMD-12 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | 1.8 | 10 | uM |
| XMD-12 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -7.1 | 10 | uM |
| XMD-12 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 22.4 | 10 | uM |
| XMD-12 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -71.5 | 10 | uM |
| XMD-12 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -17.2 | 10 | uM |
| XMD-12 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -24.3 | 10 | uM |
| XMD-12 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | 28.1 | 10 | uM |
| XMD-12 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -4.3 | 10 | uM |
| XMD-12 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | -32.7 | 10 | uM |
| XMD-12 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | 14.9 | 10 | uM |