XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | 11.2 | 10 | uM |
XMD-12 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -11.7 | 10 | uM |
XMD-12 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 10 | uM | |
XMD-12 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -20.1 | 10 | uM |
XMD-12 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -7.5 | 10 | uM |
XMD-12 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -2.6 | 10 | uM |
XMD-12 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.2 | 10 | uM |
XMD-12 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | 10 | uM | |
XMD-12 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -208.2 | 10 | uM |
XMD-12 | HeLa | TLK1 | YAAVkIHQLNK | Lys1 | -23.8 | 10 | uM |
XMD-12 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | -47.5 | 10 | uM |
XMD-12 | PC-3 | ILK | WQGIVVkVLK | Lys1 | -12.5 | 10 | uM |
XMD-12 | HeLa | ILK | WQGIVVkVLK | Lys1 | -4.0 | 10 | uM |
XMD-12 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | 11.4 | 10 | uM |
XMD-12 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 15.8 | 10 | uM |
XMD-12 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 66.5 | 10 | uM |
XMD-12 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -14.1 | 10 | uM |
XMD-12 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -23.4 | 10 | uM |
XMD-12 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.2 | 10 | uM |
XMD-12 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -5.8 | 10 | uM |
XMD-12 | HeLa | PAN3 | VMDPTkILITGK | -13.7 | 10 | uM | |
XMD-12 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -23.2 | 10 | uM |
XMD-12 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 14.4 | 10 | uM |
XMD-12 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | -11.2 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 2.2 | 10 | uM |