XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -2.6 | 10 | uM |
| XMD-12 | PC-3 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 49.7 | 10 | uM |
| XMD-12 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 14.8 | 10 | uM |
| XMD-12 | HeLa | IRAK3 | SHLEHQSCTINMTSSSSkHLWYMPEEYIR | Protein Kinase Domain | 23.7 | 10 | uM |
| XMD-12 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.2 | 10 | uM |
| XMD-12 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | -11.9 | 10 | uM |
| XMD-12 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -2.4 | 10 | uM |
| XMD-12 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -23.2 | 10 | uM |
| XMD-12 | HeLa | MK14 | QELNkTIWEVPER | Other | -2.7 | 10 | uM |
| XMD-12 | PC-3 | ROCK1 | kLQLELNQER | Other | -25.8 | 10 | uM |
| XMD-12 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 2.8 | 10 | uM |
| XMD-12 | PC-3 | MK14 | QELNkTIWEVPER | Other | -5.0 | 10 | uM |
| XMD-12 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 92.9 | 10 | uM |
| XMD-12 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 31.8 | 10 | uM |
| XMD-12 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.3 | 10 | uM |
| XMD-12 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 2.9 | 10 | uM |
| XMD-12 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 24.9 | 10 | uM |
| XMD-12 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 0.2 | 10 | uM |
| XMD-12 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | 28.1 | 10 | uM |
| XMD-12 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -16.7 | 10 | uM |
| XMD-12 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 64.7 | 10 | uM |
| XMD-12 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -6.9 | 10 | uM |
| XMD-12 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 14.3 | 10 | uM |
| XMD-12 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -16.3 | 10 | uM |
| XMD-12 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 62.7 | 10 | uM |