XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -16.1 | 10 | uM |
XMD8-92 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -15.7 | 10 | uM |
XMD8-92 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 11.8 | 10 | uM |
XMD8-92 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -7.2 | 10 | uM |
XMD8-92 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 0.1 | 10 | uM |
XMD8-92 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.5 | 10 | uM |
XMD8-92 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.5 | 10 | uM |
XMD8-92 | PC-3 | EGFR | IPVAIkELR | Lys1 | -5.4 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.0 | 10 | uM |
XMD8-92 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -20.3 | 10 | uM |
XMD8-92 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 10.8 | 10 | uM |
XMD8-92 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.0 | 10 | uM |
XMD8-92 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 54.0 | 10 | uM |
XMD8-92 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -2.2 | 10 | uM |
XMD8-92 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 5.2 | 10 | uM |
XMD8-92 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 8.9 | 10 | uM |
XMD8-92 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -26.2 | 10 | uM |
XMD8-92 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 7.6 | 10 | uM |
XMD8-92 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -8.6 | 10 | uM |
XMD8-92 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 6.7 | 10 | uM |
XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -12.5 | 10 | uM |
XMD8-92 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 1.5 | 10 | uM |
XMD8-92 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 6.0 | 10 | uM |
XMD8-92 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -28.7 | 10 | uM |