XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
-4.1
10
uM
XMD8-92 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-25.7
10
uM
XMD8-92 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
11.1
10
uM
XMD8-92 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
-9.3
10
uM
XMD8-92 HeLa SYK
ISDFGLSkALR
Activation Loop
-2.7
10
uM
XMD8-92 HeLa TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD8-92 PC-3 TLK1
YAAVkIHQLNK
Lys1
13.2
10
uM
XMD8-92 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-12.6
10
uM
XMD8-92 HeLa AurB
SHFIVALkVLFK
Lys1
9.7
10
uM
XMD8-92 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
-15.6
10
uM
XMD8-92 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
7.3
10
uM
XMD8-92 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-19.5
10
uM
XMD8-92 PC-3 SNRK
DLkPENVVFFEK
Lys2
0.3
10
uM
XMD8-92 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-50.1
10
uM