XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
7.9
10
uM
XMD8-92 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
9.2
10
uM
XMD8-92 HeLa MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
9.1
10
uM
XMD8-92 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
30.3
10
uM
XMD8-92 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
4.6
10
uM
XMD8-92 HeLa KS6B1
DLkPENIMLNHQGHVK
Lys2
-2.3
10
uM
XMD8-92 HeLa KS6B2
DLkPENIMLSSQGHIK
Lys2
-13.2
10
uM
XMD8-92 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-11.2
10
uM
XMD8-92 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
18.5
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
11.7
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-16.3
10
uM
XMD8-92 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
8.3
10
uM
XMD8-92 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
-1.4
10
uM
XMD8-92 PC-3 SNRK
DLkPENVVFFEK
Lys2
0.3
10
uM
XMD8-92 HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-13.0
10
uM
XMD8-92 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
6.1
10
uM
XMD8-92 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
-10.9
10
uM
XMD8-92 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-11.2
10
uM
XMD8-92 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-12.6
10
uM
XMD8-92 HeLa PCTAIRE2
DLkPQNLLINEK
Lys2
-24.6
10
uM
XMD8-92 PC-3 CDK5
DLkPQNLLINR
Lys2
-1.0
10
uM
XMD8-92 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
-18.6
10
uM
XMD8-92 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
9.2
10
uM
XMD8-92 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
5.1
10
uM
XMD8-92 HeLa PEK
DLkPSNIFFTMDDVVK
Lys2
-1.4
10
uM