XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 7.9 | 10 | uM |
XMD8-92 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 9.2 | 10 | uM |
XMD8-92 | HeLa | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | 9.1 | 10 | uM |
XMD8-92 | HeLa | RSK1,RSK2_domain1 | DLkPENILLDEEGHIKLTDFGLSK | Lys2 | 30.3 | 10 | uM |
XMD8-92 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 4.6 | 10 | uM |
XMD8-92 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -2.3 | 10 | uM |
XMD8-92 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -13.2 | 10 | uM |
XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 18.5 | 10 | uM |
XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
XMD8-92 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -1.4 | 10 | uM |
XMD8-92 | PC-3 | SNRK | DLkPENVVFFEK | Lys2 | 0.3 | 10 | uM |
XMD8-92 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -13.0 | 10 | uM |
XMD8-92 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | 6.1 | 10 | uM |
XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -12.6 | 10 | uM |
XMD8-92 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -24.6 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | -1.0 | 10 | uM |
XMD8-92 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -18.6 | 10 | uM |
XMD8-92 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 9.2 | 10 | uM |
XMD8-92 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 5.1 | 10 | uM |
XMD8-92 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -1.4 | 10 | uM |