XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa MLTK
WISQDKEVAVKk
Lys1
-0.8
10
uM
XMD8-92 HeLa ILK
WQGNDIVVkVLK
Lys1
-4.9
10
uM
XMD8-92 PC-3 ILK
WQGNDIVVkVLK
Lys1
17.7
10
uM
XMD8-92 HeLa TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD8-92 PC-3 TLK1
YAAVkIHQLNK
Lys1
13.2
10
uM
XMD8-92 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-18.1
10
uM
XMD8-92 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-6.2
10
uM
XMD8-92 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.5
10
uM
XMD8-92 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-5.5
10
uM
XMD8-92 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
6.9
10
uM
XMD8-92 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
3.4
10
uM
XMD8-92 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-20.9
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-50.1
10
uM