XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-9.2
10
uM
XMD8-92 PC-3 EPHA2
EVPVAIkTLK
Lys1
-10.5
10
uM
XMD8-92 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-2.0
10
uM
XMD8-92 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-5.7
10
uM
XMD8-92 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
10.7
10
uM
XMD8-92 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-3.7
10
uM
XMD8-92 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.0
10
uM
XMD8-92 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
54.0
10
uM
XMD8-92 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
5.2
10
uM
XMD8-92 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
-2.2
10
uM
XMD8-92 HeLa FES
LRADNTLVAVkSCR
Lys1
-4.8
10
uM
XMD8-92 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
8.9
10
uM
XMD8-92 HeLa GCK
DTVTSELAAVkIVK
Lys1
-26.2
10
uM
XMD8-92 PC-3 GCN2
LDGCCYAVkR
Lys1
9.4
10
uM
XMD8-92 HeLa GCN2
LDGCCYAVkR
Lys1
-5.2
10
uM
XMD8-92 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.6
10
uM
XMD8-92 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-8.6
10
uM
XMD8-92 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
6.7
10
uM
XMD8-92 HeLa HPK1
DKVSGDLVALkMVK
Lys1
-2.2
10
uM
XMD8-92 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-11.2
10
uM
XMD8-92 HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
-1.3
10
uM
XMD8-92 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
1.5
10
uM
XMD8-92 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-12.5
10
uM
XMD8-92 HeLa ILK
WQGNDIVVkVLK
Lys1
-4.9
10
uM
XMD8-92 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
6.0
10
uM