XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -9.2 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -10.5 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.0 | 10 | uM |
XMD8-92 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -5.7 | 10 | uM |
XMD8-92 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 10.7 | 10 | uM |
XMD8-92 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | -3.7 | 10 | uM |
XMD8-92 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.0 | 10 | uM |
XMD8-92 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 54.0 | 10 | uM |
XMD8-92 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 5.2 | 10 | uM |
XMD8-92 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -2.2 | 10 | uM |
XMD8-92 | HeLa | FES | LRADNTLVAVkSCR | Lys1 | -4.8 | 10 | uM |
XMD8-92 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 8.9 | 10 | uM |
XMD8-92 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -26.2 | 10 | uM |
XMD8-92 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 9.4 | 10 | uM |
XMD8-92 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -5.2 | 10 | uM |
XMD8-92 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 7.6 | 10 | uM |
XMD8-92 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -8.6 | 10 | uM |
XMD8-92 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 6.7 | 10 | uM |
XMD8-92 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -2.2 | 10 | uM |
XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -1.3 | 10 | uM |
XMD8-92 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 1.5 | 10 | uM |
XMD8-92 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -12.5 | 10 | uM |
XMD8-92 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.9 | 10 | uM |
XMD8-92 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 6.0 | 10 | uM |